BDBM16175 CHEMBL108468::UKI-1::ethyl 4-(3-carbamimidoyl-N-{[2,4,6-tris(1-methylethyl)phenyl]sulfonyl}phenylalanyl)piperazine-1-carboxylate::ethyl 4-[3-(3-carbamimidoylphenyl)-2-{[2,4,6-tris(propan-2-yl)benzene]sulfonamido}propanoyl]piperazine-1-carboxylate
SMILES CCOC(=O)N1CCN(CC1)C(=O)C(Cc1cccc(c1)C(N)=N)NS(=O)(=O)c1c(cc(cc1C(C)C)C(C)C)C(C)C
InChI Key InChIKey=ISJSHQTWOHGCMM-UHFFFAOYSA-N
Data 6 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 16175
Affinity DataKi: 37nM ΔG°: -10.1kcal/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 410nM ΔG°: -8.71kcal/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Tested for inhibition of plasminogen activator urokinase (microPa)More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Tested for inhibition of plasminMore data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nM ΔG°: -7.24kcal/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair