BDBM17004 BX-517::Indolinone based inhibitor, 4i::[(3Z)-2-oxo-3-[1-(1H-pyrrol-2-yl)ethylidene]-2,3-dihydro-1H-indol-5-yl]urea
SMILES C\C(=C1\C(=O)Nc2ccc(NC(N)=O)cc12)c1ccc[nH]1
InChI Key InChIKey=DFURSNCTQGJRRX-JYRVWZFOSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 17004
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Brigham Young University
Curated by ChEMBL
Brigham Young University
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of PDK1 (unknown origin) after 1 hr in presence of Ser/Thr-07 by fluorometric assayMore data for this Ligand-Target Pair