BDBM170444 US9085531, 14
SMILES CN1CC(c2ccc3occc3c2)c2ccccc2C1
InChI Key InChIKey=YSXLAKJPPGTIOK-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 170444
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataKi: 2nMpH: 7.4Assay Description:In order to evaluate the relative affinity of the various compounds at the NE, DA and 5HT transporters, HEK293E cell lines were developed to express ...More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMpH: 7.4Assay Description:In order to evaluate the relative affinity of the various compounds at the NE, DA and 5HT transporters, HEK293E cell lines were developed to express ...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataKi: 19.2nMpH: 7.4Assay Description:In order to evaluate the relative affinity of the various compounds at the NE, DA and 5HT transporters, HEK293E cell lines were developed to express ...More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]Nisoxetine from human NET expressed in HEK293E cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Displacement of [3H]WIN 35,428 from human DAT expressed in HEK293E cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]Citolapram from human SERT expressed in HEK293E cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair