BDBM170453 US9085531, 100
SMILES CN1CC(c2ccc3sccc3c2)c2ccc(cc2C1)N1CCOCC1
InChI Key InChIKey=QLQQUDCJVQOCBW-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 170453
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataKi: 7.10nMpH: 7.4Assay Description:In order to evaluate the relative affinity of the various compounds at the NE, DA and 5HT transporters, HEK293E cell lines were developed to express ...More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataKi: 7.60nMpH: 7.4Assay Description:In order to evaluate the relative affinity of the various compounds at the NE, DA and 5HT transporters, HEK293E cell lines were developed to express ...More data for this Ligand-Target Pair
Affinity DataKi: 53.4nMpH: 7.4Assay Description:In order to evaluate the relative affinity of the various compounds at the NE, DA and 5HT transporters, HEK293E cell lines were developed to express ...More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataIC50: 93nMAssay Description:Displacement of [125I]-RTI-55 from recombinant NET (unknown origin) expressed in HEK cells by saturation binding analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Displacement of [125I]-RTI-55 from recombinant DAT (unknown origin) expressed in HEK cells by saturation binding analysisMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Albany Molecular Research
US Patent
Albany Molecular Research
US Patent
Affinity DataIC50: 4.90nMAssay Description:Displacement of [125I]-RTI-55 from recombinant SERT (unknown origin) expressed in HEK cells by saturation binding analysisMore data for this Ligand-Target Pair