BDBM177103 US9120749, 469
SMILES CN1CCN(CC1)c1ccc(Nc2c(cnc3ccc(cc23)-c2cnc(nc2)C#N)C(=O)C2CC2)cn1
InChI Key InChIKey=OCPIPNPULRAZBD-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 177103
Affinity DataIC50: 1.5nMpH: 7.4 T: 2°CAssay Description:MELK activity was determined in the presence or absence of compounds using fluorescein isothiocyanate-labeled (FITC-labeled) histone H3 peptide as a ...More data for this Ligand-Target Pair