BDBM18619 (18Z)-12-methoxy-3,5,5-trimethyl-18-[(3-{[(2,2,2-trifluoroethyl)amino]methyl}thiophen-2-yl)methylidene]-17-oxa-6-azatetracyclo[8.8.0.0^{2,7}.0^{11,16}]octadeca-1(10),2(7),3,8,11,13,15-heptaen-13-ol::Amine, 13
SMILES COc1c(O)ccc2O\C(=C/c3sccc3CNCC(F)(F)F)c3c(ccc4NC(C)(C)C=C(C)c34)-c12
InChI Key InChIKey=OZWRZVFUZNYXMF-NHDPSOOVSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 18619
Affinity DataIC50: 0.900nM EC50: 0.5nMpH: 7.5Assay Description:GR-Mediated Agonist Activity Assay- GR-mediated activation by compounds is measured against maximal activation of dexamethasone in the same experimen...More data for this Ligand-Target Pair