BDBM194781 US9206167, 2::USRE48059, Compound of Example 2
SMILES O=c1[nH]c2ccccc2cc1OCCN1CCN(CC1)c1cccc2sccc12
InChI Key InChIKey=BOKAVZYMEBZBJT-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 194781
Affinity DataKi: 1.5nMAssay Description:5-HT2A: The binding assay was performed using 40 μl of the membrane specimen, 20 μl of [3H]-Ketanserin (final concentration 1 to 3 nM), 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nM ΔG°: -12.5kcal/molepH: 7.4 T: 2°CAssay Description:The assay was performed according to the method by Leysen J E et al. (Leysen J E, Niemegeers C J E, Van Nueten J M and Laduron P M. [3H] Ketanserin (...More data for this Ligand-Target Pair