BDBM195569 (2E)-2-[(5-Bromofuran-2-yl)methylidene]-5-methoxy-2,3-dihydro-1H-inden-1-one (11o)
SMILES COc1ccc2C(=O)\C(Cc2c1)=C\c1ccc(Br)o1
InChI Key InChIKey=UJKXUNOFSDTDGU-CSKARUKUSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 195569
Affinity DataIC50: 183nMpH: 7.4Assay Description:Recombinant human MAO-A and MAO-B were used for these studies and
kynuramine served as enzyme substrate. Kynuramine is oxidised by both
MAO isoform...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMpH: 7.4Assay Description:Recombinant human MAO-A and MAO-B were used for these studies and
kynuramine served as enzyme substrate. Kynuramine is oxidised by both
MAO isoform...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human MAO-B assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as substrate incubated for 20 mins by f...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human MAO-A assessed as inhibition of 4-hydroxyquinoline formation using kynuramine as substrate incubated for 20 mins by f...More data for this Ligand-Target Pair