BDBM195657 US9206173, 2419
SMILES COc1ccc(C(=O)N2CCc3nc(NC(C)c4ccc(cc4)C(F)(F)F)n(OC)c(=O)c3C2)c(OC)n1
InChI Key InChIKey=WSDFAEVOFGBGJE-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 195657
Affinity DataKi: 7nM ΔG°: -11.1kcal/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
Affinity DataIC50: 228nMpH: 7.4 T: 2°CAssay Description:HEK293 cells expressing human GPR10 were maintained in Dulbecco's Modified Eagles' medium supplemented with 10% fetal bovine serum, 1% penici...More data for this Ligand-Target Pair