BDBM195668 US9206173, 2430
SMILES COn1c(NC(C)c2ccc(Cl)cc2)nc2CCN(Cc2c1=O)C(=O)COc1ccc(Cl)cc1
InChI Key InChIKey=JAICWKJMHDECAE-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 195668
Affinity DataKi: 15nM ΔG°: -10.7kcal/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMpH: 7.4 T: 2°CAssay Description:HEK293 cells expressing human GPR10 were maintained in Dulbecco's Modified Eagles' medium supplemented with 10% fetal bovine serum, 1% penici...More data for this Ligand-Target Pair