BDBM195689 US9206173, 2451
SMILES CCOc1ccc(cc1)C(=O)N1CCc2nc(NC(C)c3ccc(cc3)C(F)(F)F)n(OC)c(=O)c2C1
InChI Key InChIKey=WZVABFGIISCZFI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 195689
Affinity DataKi: 9nM ΔG°: -11.0kcal/molepH: 7.4 T: 2°CAssay Description:Receptor-expressing HEK 293 cell membrane fraction was analyzed by modifying the methods of C. J. Langmead et al. (see Langmead C J, Szekeres P G; Ch...More data for this Ligand-Target Pair
Affinity DataIC50: 1.29E+3nMpH: 7.4 T: 2°CAssay Description:HEK293 cells expressing human GPR10 were maintained in Dulbecco's Modified Eagles' medium supplemented with 10% fetal bovine serum, 1% penici...More data for this Ligand-Target Pair