BDBM202494 US9238651, A55
SMILES CC(C)n1cc(cn1)-c1cnc2[nH]cc(-c3cc(nc(N)n3)C(C)(O)c3ccccc3)c2c1
InChI Key
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 202494
Affinity DataIC50: 492nMpH: 8.0 T: 2°CAssay Description:The cellular assay for the determination of the PDK1 kinase activity is
carried out as a Luminex assay in the 96-well format. PC3 cells are sown
at...More data for this Ligand-Target Pair
Affinity DataIC50: 54nMT: 2°CAssay Description:The experimental batches are carried out in a flashplate system with 384 wells/microtitration plate.In each case, the PDK1 sample His6-PDK1(Δ1-...More data for this Ligand-Target Pair