BDBM20345 3-{[4-(azepan-1-yl)phenyl]methyl}-1-(3-methylisoquinolin-5-yl)urea::Isoquinoline Analogue, 39
SMILES Cc1cc2c(NC(=O)NCc3ccc(cc3)N3CCCCCC3)cccc2cn1
InChI Key InChIKey=CRXMYQXPWMGLMV-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 20345
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Abbott Laboratories
Abbott Laboratories
Affinity DataEC50: 3.80nMpH: 7.4 T: 2°CAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair