BDBM204862 EA2/MRS5811::US9227979, 11
SMILES Cn1cc2c(n1)nc(NC(=O)Nc1ccc(CC(O)=O)cc1)n1nc(nc21)-c1ccco1
InChI Key InChIKey=QOVZGPDUOLJANP-UHFFFAOYSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 204862
TargetAdenosine receptor A3(Homo sapiens (Human))
The United States of America, As Represented By The Secretary, Department of Health and Human Services
US Patent
The United States of America, As Represented By The Secretary, Department of Health and Human Services
US Patent
Affinity DataKi: 128nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
The United States of America, As Represented By The Secretary, Department of Health and Human Services
US Patent
The United States of America, As Represented By The Secretary, Department of Health and Human Services
US Patent
Affinity DataKi: 128nMAssay Description:Displacement of [125I]AB-MEC from recombinant human A3R expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Displacement of [3H]CGS21680 from recombinant human A2AAR expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair