BDBM204958 US9249085, I(r)::US9624159, Compound I(r)
SMILES OC(=O)COc1ccc(Cl)c(NCc2cc(ccc2F)-c2cccc(F)c2)c1Cl
InChI Key InChIKey=YPQKUWFLQHVMFG-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 204958
Affinity DataEC50: 45nMAssay Description:Human CHO cells expressing the recombinant human prostanoid EP2 receptor were suspended in assay medium (HBSS buffer (Invitrogen) containing 20 mM HE...More data for this Ligand-Target Pair
Affinity DataIC50: >300nMAssay Description:Cell membrane homogenate from Human embryonic kidney HEK-293(T) cells expressing recombinant human prostanoid EP4 receptor was used to perform Prosta...More data for this Ligand-Target Pair
Affinity DataIC50: >300nMpH: 6.0Assay Description:The competition reaction was initiated by incubation of membrane protein homogenate (20 μg protein) for 120 min at 22° C. with 0.5 nM [3H]PGE2 l...More data for this Ligand-Target Pair