BDBM20641 methyl 4-[(5-carbamoyl-2-methylphenyl)amino]-5-methylpyrrolo[1,2-a][1,2,4]triazine-6-carboxylate::pyrrolo[2,1-f][1,2,4]triazine analogue, 3c

SMILES COC(=O)c1cn2ncnc(Nc3cc(ccc3C)C(N)=O)c2c1C

InChI Key InChIKey=ZDGDOXAQILZWIJ-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20641   

TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM20641(methyl 4-[(5-carbamoyl-2-methylphenyl)amino]-5-met...)
Affinity DataIC50:  78nM EC50: >2.00E+3nMpH: 7.5 T: 2°CAssay Description:The kinase activity was determined by quantitation of the amount of radioactive phosphate transferred to myelin basic protein (MBP) with or without i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed