BDBM210752 US9290454, 3.4
SMILES C[C@@H](NC(=O)c1ccc2c(cc(CCCCC(O)=O)n(-c3ccc(cc3)C#N)c2=O)c1)c1ccc(F)cc1
InChI Key InChIKey=GERCAPRDMLSXBV-LJQANCHMSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 210752
Affinity DataKi: 8.84nM ΔG°: -11.9kcal/molepH: 7.4 T: 2°CAssay Description:Radioligand binding was performed using filtration or scintillation proximity assay (SPA) technology. SPA assays were done at room temperature in 10 ...More data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Antagonist activity at human CRTh2 expressed in HEK cells assessed as inhibition of DK-PGD2-mediated attenuation of forskolin-induced cAMP accumulati...More data for this Ligand-Target Pair