BDBM210903 US9273043, A158(a)
SMILES C[C@H]1CN(CCN1C(=O)Nc1nc2cc(F)c(F)cc2s1)c1ncc(cc1F)[C@H](O)CO
InChI Key InChIKey=PLPNXVMXQNODJV-MGPLVRAMSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 210903
Affinity DataIC50: 17.1nMpH: 7.2 T: 37°CAssay Description:pH dependent Ca2+ responses in TRPV1/CHO cells cultured in a 96-well plate were determined (see, e.g., FIG. 2 of U.S. Patent Application Publication ...More data for this Ligand-Target Pair
Affinity DataIC50: 62.4nMpH: 7.4Assay Description:One day prior to assay, TRPV1/CHO cells were seeded in 96-well clear-bottom black plates (20,000 cells/well) in growth media. On the day of the exper...More data for this Ligand-Target Pair