BDBM237479 US9393232, 2.57a::US9393232, 2.57b
SMILES Cc1noc(C)c1-c1ccc2NC(=O)C(N[C@H](CO)Cc3cnc[nH]3)(c2c1)c1ccccc1
InChI Key
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 237479
Affinity DataIC50: 41nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Affinity DataIC50: 410nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair