BDBM237516 US9393232, 2.17::US9393232, 2.17a::US9393232, 2.17b
SMILES Cc1noc(C)c1-c1ccc2NC(=O)C(N3CCC[C@@H](O)C3)(c2c1)c1ccccc1
InChI Key InChIKey=UXFXOEGGFKVCDW-PHSANKKPSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 237516
Affinity DataIC50: 40nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMpH: 7.5Assay Description:The assay was carried out in binding mixtures of the bromodomain protein, 0-10 μM compounds and tetra-acetylated histone peptide (SGRGAC.KGGAC.K...More data for this Ligand-Target Pair