BDBM239860 US9403767, 9
SMILES CNC1(CCC(CC1)(N(C)C)c1ccccc1)c1ccccc1
InChI Key InChIKey=FAOUSJRZQIHJRX-UHFFFAOYSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 239860
Affinity DataKi: 17.8nMpH: 7.4Assay Description:The compounds were examined with membranes of recombinant CHO-ORL 1 cells in a receptor binding assay with 3H-nociceptin/orphanin FQ. This test syste...More data for this Ligand-Target Pair
Affinity DataKi: 640nM ΔG°: -8.44kcal/moleT: 2°CAssay Description:The affinity to the human μ-opiate receptor was determined in a homogeneous preparation in microtiter plates. For this, dilution series of the res...More data for this Ligand-Target Pair
Affinity DataKi: 1.17E+3nM ΔG°: -8.09kcal/moleT: 2°CAssay Description:The determination occurred in a homogeneous batch in microtiter plates. For this, dilution series of the respective substances to be tested were incu...More data for this Ligand-Target Pair