BDBM242438 US9422235, 12
SMILES COc1cc(Nc2ccc(cc2)S(=O)(=O)NCC2CC2)cc(OC)c1
InChI Key InChIKey=GCPFDXOLQNQCTI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 242438
Affinity DataKi: 6nM ΔG°: -11.4kcal/mole IC50: 11nMT: 2°CAssay Description:The binding assays were performed by testing the ability of the new compounds to displace the radiolabeled synthetic non-selective cannabinoid agonis...More data for this Ligand-Target Pair
Affinity DataKi: 97nM ΔG°: -9.72kcal/mole IC50: 235nMT: 2°CAssay Description:The binding assays were performed by testing the ability of the new compounds to displace the radiolabeled synthetic non-selective cannabinoid agonis...More data for this Ligand-Target Pair
Affinity DataKi: 363nM ΔG°: -8.93kcal/mole IC50: 853nMT: 2°CAssay Description:The binding assays were performed by testing the ability of the new compounds to displace the radiolabeled synthetic non-selective cannabinoid agonis...More data for this Ligand-Target Pair
Affinity DataKi: 2.68E+3nM ΔG°: -7.72kcal/mole IC50: 6.00E+3nMT: 2°CAssay Description:The binding assays were performed by testing the ability of the new compounds to displace the radiolabeled synthetic non-selective cannabinoid agonis...More data for this Ligand-Target Pair
Affinity DataKi: 2.68E+3nM ΔG°: -7.72kcal/mole IC50: 6.00E+3nMT: 2°CAssay Description:The binding assays were performed by testing the ability of the new compounds to displace the radiolabeled synthetic non-selective cannabinoid agonis...More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nM ΔG°: -7.66kcal/moleT: 2°CAssay Description:The binding assays were performed by testing the ability of the new compounds to displace the radiolabeled synthetic non-selective cannabinoid agonis...More data for this Ligand-Target Pair
Affinity DataKi: 5.56E+3nM ΔG°: -7.28kcal/mole IC50: 1.10E+4nMT: 2°CAssay Description:The binding assays were performed by testing the ability of the new compounds to displace the radiolabeled synthetic non-selective cannabinoid agonis...More data for this Ligand-Target Pair