BDBM246464 US9447114, 25
SMILES Cc1c(sc2n(C)c(=O)n(CCCO)c(=O)c12)-c1ccc(Cl)cc1
InChI Key InChIKey=WQRGHSSPNYUZEW-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 246464
Affinity DataIC50: 15.7nMpH: 7.2Assay Description:TRPC5 cells were induced 20-48 hours, removed from growth plates, and replated at low density (to attain good single-cell physical separation) on gla...More data for this Ligand-Target Pair
Affinity DataIC50: 168nMpH: 7.4 T: 2°CAssay Description:The commercially available HEK293/TREx line (Invitrogen) was stably transfected with a TRPC5 construct and screened by conventional calcium imaging t...More data for this Ligand-Target Pair