BDBM263553 2-{5-amino-1-[2-chloro-4-(3- cyano-phenoxy)-phenyl]-1h- pyrazole-4-carbonyl}-n-cyano- 1h-indole-5-carboxylic acid amide::US9556150, i-41
SMILES Nc1c(cnn1-c1ccc(Oc2cccc(c2)C#N)cc1Cl)C(=O)c1cc2cc(ccc2[nH]1)C(=O)NC#N
InChI Key InChIKey=DWFZKHPBAFWVNS-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 263553
Affinity DataIC50: 52nMpH: 7.15Assay Description:This BTK competition assay measures compound potency (IC50) for the inactivated state of Bruton's Tyrosine Kinase using FRET (Förster/Fluorescenc...More data for this Ligand-Target Pair