BDBM264120 3-(4-(4-(4-(4-oxofuro[3,2-c]pyridin-5 (4H)-yl)phenyl)piperazin-1-yl)butyl)-1H-indole-5-carbonitrile::US9714232, 33
SMILES O=c1n(ccc2occc12)-c1ccc(cc1)N1CCN(CCCCc2c[nH]c3ccc(cc23)C#N)CC1
InChI Key InChIKey=RLGFCRXXEKJBKA-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 264120
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Sunshine Lake Pharma
Curated by ChEMBL
Sunshine Lake Pharma
Curated by ChEMBL
Affinity DataIC50: 0.530nMAssay Description:Inhibition of serotonin transporter expressed in rat brain tissue assessed as inhibition of [3H]-5-hydroxytryptamine reuptake measured after 15 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of 5-HT3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of 5-HT2a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of 5-HT2c (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibition of 5-HT1a (unknown origin)More data for this Ligand-Target Pair