BDBM267777 4-(4-amino-7-chloro-1-{(3R)-1-[(3-methyloxetan-3-yl)carbonyl]piperidin-3-yl}-1H-pyrazolo[4,3-c]pyridin-3-yl)-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide::US9718828, Example, 383
SMILES COCC(=O)N1CCC[C@H](C1)n1nc(-c2ccc(cc2)C(=O)Nc2cc(ccn2)C(F)(F)F)c2c(N)nccc12
InChI Key InChIKey=SEBXNLHOPSBRNT-LJQANCHMSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 267777
Affinity DataIC50: <10nMAssay Description:BTK enzymatic activity was determined with the LANCE (Lanthanide Chelate Excite) TR-FRET (Time-resolved fluorescence resonance energy transfer) assay...More data for this Ligand-Target Pair