BDBM272134 (R)-2-(1,3-Dimethyl-1H-pyrazol-5-yl)-5-(3-fluoro-2- methylphenyl)-N-hydroxy-5,6-dihydro-4H- cyclopenta[d]thiazole-5-carboxamide::US10065948, 70::US10457675, Example 70

SMILES Cc1cc(-c2nc3C[C@](Cc3s2)(C(=O)NO)c2cccc(F)c2C)n(C)n1

InChI Key InChIKey=GABUTZUDMAPMJE-LJQANCHMSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 272134   

TargetHistone deacetylase 9(Homo sapiens (Human))
Chdi Foundation

US Patent
LigandPNGBDBM272134((R)-2-(1,3-Dimethyl-1H-pyrazol-5-yl)-5-(3-fluoro-2...)
Affinity DataIC50:  122nMAssay Description:The potency of the compounds is quantified by measuring the Histone Deacetylase 9 (HDAC9) enzymatic activity using the fluorogenic substrate, Boc-Lys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 9(Homo sapiens (Human))
Chdi Foundation

US Patent
LigandPNGBDBM272134((R)-2-(1,3-Dimethyl-1H-pyrazol-5-yl)-5-(3-fluoro-2...)
Affinity DataIC50:  122nMAssay Description:The potency of the compounds is quantified by measuring the Histone Deacetylase 9 (HDAC9) enzymatic activity using the fluorogenic substrate, Boc-Lys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent