BDBM273029 N-{(R)-1-[5-(1-chlorocyclopropyl)-7-oxo-6,7-dihydro[1,3]thiazolo[5,4-d]pyrimidin-2-yl]ethyl}-N-methylcarbamic acid phenyl ester::US10065972, Example 85
SMILES C[C@@H](N(C)C(=O)Oc1ccccc1)c1nc2c(nc([nH]c2=O)C2(Cl)CC2)s1
InChI Key InChIKey=MMLNMAREBGQISI-SNVBAGLBSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 273029
TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Homo sapiens (Human))
Mitsubishi Tanabe Pharma
US Patent
Mitsubishi Tanabe Pharma
US Patent
Affinity DataIC50: 170nMpH: 8.0Assay Description:The inhibitory action of the test compound on human recombinant KAT-II was determined by the following method.To a reaction mixture (45 μL) cont...More data for this Ligand-Target Pair