BDBM274546 N-(6-(4-(4-fluorophenyl)-1- (1-(3,3,3-trifluoropropanoyl) piperidin-4-yl)-1H- imidazol-5-yl)imidazo[1,2-b] pyridazin-2-yl)thiazole- 5-carboxamide::US9556179, Compound 117
SMILES Fc1ccc(cc1)-c1ncn(C2CCN(CC2)C(=O)CC(F)(F)F)c1-c1ccc2nc(NC(=O)c3cncs3)cn2n1
InChI Key InChIKey=SDQBTGBRICOINB-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 274546
Affinity DataIC50: 0.175nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Affinity DataIC50: 0.424nMpH: 7.4 T: 2°CAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair