BDBM278827 2-(1,4-diazepan-1-yl)- N-[1-methyl-3- (trifluoromethyl)-1H- pyrazol-4-yl] thieno[2,3-b] pyrazine-7- carboxamide::US10040802, Example 6
SMILES Cn1cc(NC(=O)c2csc3ncc(nc23)N2CCCNCC2)c(n1)C(F)(F)F
InChI Key InChIKey=OLTBSNVUBBDTIX-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 278827
Affinity DataIC50: 17nMpH: 7.2Assay Description:The kinase activity of IRAK4 is determined by its ability to catalyze the phosphorylation of a fluorescent polypeptide substrate. The extent of phosp...More data for this Ligand-Target Pair