BDBM278853 4-{8-amino-3- [(6S,8aR)-6-methyl-3- oxohexahydro[1,3] oxazolo[3,4-a]pyridin- 6-yl]limidazo[1,5-a] pyrazin-1-yl}-3- ethoxy-N-[4- (trifluoromethyl) pyridin-2-yl] benzamide::US10040805, Example 1
SMILES CCOc1cc(ccc1-c1nc(n2ccnc(N)c12)[C@@]1(C)CC[C@@H]2COC(=O)N2C1)C(=O)Nc1cc(ccn1)C(F)(F)F
InChI Key InChIKey=HZBFBSZOVNDXHC-WRHNGFHOSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 278853
Affinity DataIC50: 0.610nMAssay Description:BTK enzymatic activity was determined with the LANCE (Lanthanide Chelate Excite) TR-FRET (Time-resolved fluorescence resonance energy transfer) assay...More data for this Ligand-Target Pair