BDBM278904 2-[(3R)-3- aminopiperidin- 1-yl]-N-(2- cyanophenyl)- thieno[2,3-b]- pyrazine-7- carboxamide trifluoroacetate::US10040802, Example 84
SMILES OC(=O)C(F)(F)F.N[C@@H]1CCCN(C1)c1cnc2scc(C(=O)Nc3ccccc3C#N)c2n1
InChI Key InChIKey=QOKWBEPHJZVKLK-BTQNPOSSSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 278904
Affinity DataIC50: 33nMpH: 7.2Assay Description:The kinase activity of IRAK4 is determined by its ability to catalyze the phosphorylation of a fluorescent polypeptide substrate. The extent of phosp...More data for this Ligand-Target Pair