BDBM285636 4-[3-Methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy]-1H-imidazo[4,5-c]pyridine (2)::US10077272, Example 2::US9868744, 11

SMILES Cc1cc(Oc2nccc3[nH]cnc23)ccc1-c1c(C)ncnc1C

InChI Key InChIKey=WSMJDTNHHKPQKW-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 285636   

TargetD(1A) dopamine receptor(Homo sapiens (Human))
Pfizer

US Patent
LigandPNGBDBM285636(4-[3-Methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)...)
Affinity DataKi:  374nMpH: 7.4Assay Description:D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Pfizer

US Patent
LigandPNGBDBM285636(4-[3-Methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)...)
Affinity DataKi:  912nMAssay Description:D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent