BDBM285650 4,6-dimethyl-5-{2-methyl-4-[(3-methyl[1,2]oxazolo[4,5-c]pyridin-4-yl)oxy]phenyl}pyridazin-3(2H)-one, trifluoroaceticacid salt::US10077272, Example 16::US9868744, 16

SMILES Cc1noc2ccnc(Oc3ccc(c(C)c3)-c3c(C)n[nH]c(=O)c3C)c12

InChI Key InChIKey=PSBABCDASJNITB-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 285650   

TargetD(1A) dopamine receptor(Homo sapiens (Human))
Pfizer

US Patent
LigandPNGBDBM285650(4,6-dimethyl-5-{2-methyl-4-[(3-methyl[1,2]oxazolo[...)
Affinity DataKi:  326nMAssay Description:D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Pfizer

US Patent
LigandPNGBDBM285650(4,6-dimethyl-5-{2-methyl-4-[(3-methyl[1,2]oxazolo[...)
Affinity DataKi:  326nMpH: 7.4Assay Description:D1 binding assays were performed using over-expressing LTK human cell lines. To determine basic assay parameters, ligand concentrations were determin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent