BDBM288222 7-Chloro-5-(2-cyclopropyl-6-(trifluoromethyl)-[1,2,4]triazolo[1,5-::US10087185, Example 40
SMILES FC(F)(F)c1ccc2nc(nn2c1-c1cc2CC(=O)Nc2c(Cl)c1)C1CC1
InChI Key InChIKey=NVZXOVFLBHVNJQ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 288222
TargetVoltage-dependent calcium channel gamma-8 subunit(Homo sapiens (Human))
Janssen Pharmaceutica
US Patent
Janssen Pharmaceutica
US Patent
Affinity DataIC50: 0.398nMpH: 7.4Assay Description:This assay was used to test compounds for their ability to inhibit TARP γ8 dependent AMPA receptor activity. The AMPA receptor is a non-selectiv...More data for this Ligand-Target Pair