BDBM298354 US10124003, Ex. Compound 16

SMILES COc1cc(OC)cc(c1)C#Cc1nn(C2CN(C2)C(O)\C=C\CNC2CCC2)c2ncnc(N)c12

InChI Key InChIKey=IYBYGJHPOOXALO-QPJJXVBHSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 298354   

TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM298354(US10124003, Ex. Compound 16)
Affinity DataIC50:  3.80nMAssay Description:When setting conditions for the measurement of the inhibitory effect of the compounds on FGFR2 kinase activity, FL-Peptide 22 (Caliper Life Sciences,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent