BDBM300562 3-{[(4-methylpiperazin-1-yl)acetyl]amino}-N-(5-phenylpyridin-2-yl)-4-(trifluoromethoxy)benzamide formiate::US10130633, Example 132
SMILES CC1CCN(CC(=O)Nc2cc(ccc2OC(F)(F)F)C(=O)Nc2ccc(cn2)-c2ccccc2)CC1
InChI Key InChIKey=CMAIWNCQGOARKU-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 300562
Affinity DataIC50: 35.5nMAssay Description:In preparation of the assay, the two cell lines were plated 24 hours before at 10000 cells per well of a 384 micro titre plate (MTP) in 30 μL gr...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:HEK293 cells were cotransfected with the FOP control vector and pcDNA3. The FOP vector is identical to the TOP construct, but it contains instead of ...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:In preparation of the assay, the two cell lines were plated 24 hours before beginning the test at 10000 cells per well in a 384 micro titre plate (MT...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:In preparation of the assay, the two cell lines were plated 24 hours before at 10000 cells per well of a 384 micro titre plate (MTP) in 30 μL gr...More data for this Ligand-Target Pair