BDBM317631 2-{5-Amino- 1-[4-(3-cyano- phenoxy)-2- methyl- phenyl]-1H- pyrazole-4- carbonyl}-1H- indole-4- carboxylic acid methylamide::US10640491, Compound 21::US11104668, Compound 21::US9624201, Compound 21
SMILES CNC(=O)c1cccc2[nH]c(cc12)C(=O)c1cnn(c1N)-c1ccc(Oc2cccc(c2)C#N)cc1C
InChI Key InChIKey=QWWSDFMIXCJUAQ-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 317631
Affinity DataIC50: 13nMAssay Description:The assay is a capture of radioactive 33P phosphorylated product through filtration. The interactions of Btk, biotinylated SH2 peptide substrate (Src...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:This BTK competition assay measures compound potency (IC50) for the inactivated state of Bruton's Tyrosine Kinase using FRET (Förster/Fluorescenc...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:This BTK competition assay measures compound potency (IC50) for the inactivated state of Bruton's Tyrosine Kinase using FRET (Förster/Flouresence...More data for this Ligand-Target Pair