BDBM367615 Methyl N-[(1S)-2-[4-[2-(4-amino-6-chloro-2-methyl-pyrimidin-5-yl)ethyl]-1-piperidyl]-1-methyl-2-oxo-ethyl]carbamate::US10227310, Example 71
SMILES COC(=O)N[C@@H](C)C(=O)N1CCC(CCc2c(N)nc(C)nc2Cl)CC1
InChI Key InChIKey=CTAGBUIPLIEQID-JTQLQIEISA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 367615
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 149nMAssay Description:Inhibition of human His-tagged GOAT expressed in baculovirus infected Sf9 cell membrane using desacyl-ghrelin-biotin and octanoyl-CoA as substrate in...More data for this Ligand-Target Pair
TargetGhrelin O-acyltransferase(Homo sapiens (Human))
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse And Alcoholism
Curated by ChEMBL
Affinity DataIC50: 149nMAssay Description:Prepare test compounds in DMSO to make up a 0.2 mM stock solution. Serially dilute the stock solution in DMSO for ten concentrations with final compo...More data for this Ligand-Target Pair