BDBM374606 N-{3-[3-amino-7-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-5-yl]-2-methylphenyl}-4-tert-butyl-2-fluorobenzamide::US10246457, Example 15
SMILES Cc1c(NC(=O)c2ccc(cc2F)C(C)(C)C)cccc1-c1cc(-c2cnn(C)c2)c2[nH]nc(N)c2c1
InChI Key InChIKey=YOLUQGAOJAKUDF-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 374606
Affinity DataIC50: 1.00E+3nMAssay Description:Btk enzymatic activity was determined with the LANCE (Lanthanide Chelate Excite) TR-FRET (lime-resolved fluorescence resonance energy transfer) assay...More data for this Ligand-Target Pair
Affinity DataIC50: 23.8nMAssay Description:Btk enzymatic activity was determined with the LANCE (Lanthanide Chelate Excite) TR-FRET (lime-resolved fluorescence resonance energy transfer) assay...More data for this Ligand-Target Pair