BDBM387353 2-(methylsulfanyl)-4-(4-{1H-pyrrolo[3,2-c]pyridin-1-yl}pyrrolo[2,1-f][1,2,4]triazin-2-yl)pyrimidine::US10292985, Example 35
SMILES CSc1nccc(n1)-c1nc(-n2ccc3cnccc23)c2cccn2n1
InChI Key InChIKey=XBQVOWNWPIYUND-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 387353
Affinity DataIC50: 2.20nMAssay Description:Assays are conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGFβR1 T204D or HIS-TGFβR2 WT, anti-HIS detec...More data for this Ligand-Target Pair