BDBM400284 US10328074, Example III-47
SMILES CNc1nc(cn2c(C)nnc12)-c1nc2cnc(cc2n1[C@@H](C)c1cccnc1)N1CCN(C)CC1
InChI Key InChIKey=UNZXRKWMYMYRFN-INIZCTEOSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 400284
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Boehringer Ingelheim International
US Patent
Boehringer Ingelheim International
US Patent
Affinity DataIC50: 12nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair