BDBM400991 US10005735, Compound 4
SMILES Sc1cccc2cc(cnc12)C(=O)Nc1ncco1
InChI Key InChIKey=MHBKHYFBZCYHNI-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 400991
Target26S proteasome non-ATPase regulatory subunit 14(Homo sapiens (Human))
California Institute of Technology
US Patent
California Institute of Technology
US Patent
Affinity DataIC50: 2.60E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair
TargetCOP9 signalosome complex subunit 5(Homo sapiens (Human))
California Institute of Technology
US Patent
California Institute of Technology
US Patent
Affinity DataIC50: 1.50E+4nMAssay Description:In brief, this Rpn11 bioassay employs a fluorescent polarization readout based on the ability of the 26S proteasome to cleave the protein substrate i...More data for this Ligand-Target Pair