BDBM404533 (R)-N-(1- cyanopyrrolidin- 3-yl)-2-fluoro-4- (imidazo[1,2- a]pyrazin-3- yl)benzamide::US10343992, Example 185::US10689345, Example 185::US11066365, Example 185::US11390584, Example 185
SMILES Fc1cc(ccc1C(=O)N[C@@H]1CCN(C1)C#N)-c1cnc2cnccn12
InChI Key InChIKey=HCOIOBMSMDOIFA-CYBMUJFWSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 404533
Affinity DataIC50: <100nMAssay Description:Dilution plates were prepared at 21 times the final concentration (2100 μM for a final concentration of 100 μM) in 50% DMSO in a 96-well po...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Dilution plates were prepared at 21 times the final concentration (2100 μM for a final concentration of 100 μM) in 50% DMSO in a 96-well po...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:USP30 biochemical fluorescence intensity IC50 assay Dilution plates were prepared at 21 times the final concentration (2100 μM for a final conce...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:USP30 Biochemical Fluorescence Intensity Kinetic Assay.Reactions were performed in duplicate in black 384 well plates (small volume, Greiner 784076) ...More data for this Ligand-Target Pair