BDBM426074 1-[4-[2-(4-Fluorophenyl)-3-(1H-indazol-5-yl)imidazo[1,2-a]pyrazin-8-::US10513523, Example 13
SMILES CC(=O)N1CCN(CC1)c1nccn2c(c(nc12)-c1ccc(F)cc1)-c1ccc2[nH]ncc2c1
InChI Key InChIKey=YODZKYDOJLDGMV-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 426074
Affinity DataIC50: 0.200nMAssay Description:This assay was used to test compounds for their ability to inhibit TARP γ8 dependent AMPA receptor activity. The AMPA receptor is a non-selectiv...More data for this Ligand-Target Pair