BDBM426178 6-[2-(4-Fluorophenyl)-8-morpholino-imidazo[1,2-a]pyrazin-3-yl]-3H-1,3-::US10513523, Example 118
SMILES Fc1ccc(cc1)-c1nc2c(nccn2c1-c1ccc2[nH]c(=O)sc2c1)N1CCOCC1
InChI Key InChIKey=UCUCEYHJSPWSPI-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 426178
Affinity DataIC50: 0.320nMAssay Description:This assay was used to test compounds for their ability to inhibit TARP γ8 dependent AMPA receptor activity. The AMPA receptor is a non-selectiv...More data for this Ligand-Target Pair