BDBM434903 4'-(1-(2-benzylpiperidine-1- carbonyl)-1H-1,2,3-triazol-4-yl)- N,N-dimethyl-[1,1'-biphenyl]-2- carboxamide::US10583137, Compound 77

SMILES CN(C)C(=O)c1ccccc1-c1ccc(cc1)-c1cn(nn1)C(=O)N1CCCCC1Cc1ccccc1

InChI Key InChIKey=PAQKWNYAUNFUGU-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 434903   

TargetDiacylglycerol lipase-beta(Homo sapiens (Human))
The Scripps Research Institute

US Patent
LigandPNGBDBM434903(4'-(1-(2-benzylpiperidine-1- carbonyl)-1H-1,2,3-tr...)
Affinity DataIC50:  1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
The Scripps Research Institute

US Patent
LigandPNGBDBM434903(4'-(1-(2-benzylpiperidine-1- carbonyl)-1H-1,2,3-tr...)
Affinity DataIC50: <400nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent