BDBM437293 5-(1-(1-(2-methoxyphenyl)ethyl)-1H-pyrazol-4-yl)- 1-methylpyridin-2(1H)-one::US10617680, Example 27::US11020380, Example 27

SMILES COc1ccccc1C(C)n1cc(cn1)-c1ccc(=O)n(C)c1

InChI Key InChIKey=JLGHOSWJLRBWJK-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437293   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437293(5-(1-(1-(2-methoxyphenyl)ethyl)-1H-pyrazol-4-yl)- ...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437293(5-(1-(1-(2-methoxyphenyl)ethyl)-1H-pyrazol-4-yl)- ...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent