BDBM437299 2-methyl-4-(1-(1-phenylethyl)-1H-pyrazol-4-yl)- 2,5,6,7-tetrahydro-1H-cyclopenta[c]pyridin-1-one::US10617680, Example 33::US11020380, Example 33

SMILES CC(c1ccccc1)n1cc(cn1)-c1cn(C)c(=O)c2CCCc12

InChI Key InChIKey=MNYBCXOBUOYSLQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437299   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437299(2-methyl-4-(1-(1-phenylethyl)-1H-pyrazol-4-yl)- 2,...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437299(2-methyl-4-(1-(1-phenylethyl)-1H-pyrazol-4-yl)- 2,...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent