BDBM437300 1,3-dimethyl-5-(5-methyl-1-(1-phenylethyl)-1H- pyrazol-4-yl)pyridin-2(1H)-one::US10617680, Example 34::US11020380, Example 34

SMILES CC(c1ccccc1)n1ncc(c1C)-c1cc(C)c(=O)n(C)c1

InChI Key InChIKey=QVWGIJIAGXMSIF-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437300   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437300(1,3-dimethyl-5-(5-methyl-1-(1-phenylethyl)-1H- pyr...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437300(1,3-dimethyl-5-(5-methyl-1-(1-phenylethyl)-1H- pyr...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent